Acolbifene ID:1517
| Synonyms: |
| CAS NO : 182167-02-8 |
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| Molecular Formula: C29H31NO4 |
| Molecular Weight: 457.56074 |
| Purity: 98% |
| Solubility: In DMSO |
| Storage: -20°C |
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Remarks:Acolbifene, also known as EM-652, or SCH-57068, is a selective estrogen receptor modulator (SERM). Acolbifene is currently being studied in the prevention of breast cancer in women at high risk of breast cancer. EM-652 (SCH 57068) and the prodrug EM-800 (SCH57050) which are the most potent of the known antiestrogens. EM-652 is the compound having the highest affinity for the estrogen receptor, including estradiol. It has higher affinity for the ER than ICI 182780, hydroxytamoxifen, raloxifene, droloxifene and hydroxytoremifene. EM-652 has the most potent inhibitory activity on both ER alpha and ER beta compared to any of the other antiestrogens tested. EM-652 was also the most potent inhibitor of the percentage of cycling cancer cells.
Quality Control
H-NMR,C-NMR,LC-MS,HPLC. |
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