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Cas No. |
Product name |
934526-89-3 |
Pilaralisib (XL147) |
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Pilaralisib (XL147) is a selective and reversible class I PI3K inhibitor for PI3Kα/δ/γ with IC50 of 39 nM/36 nM/23 nM in cell-free assays, less potent to PI3Kβ. Phase 1/2. |
755038-65-4 |
Volasertib(BI6727) |
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Volasertib (BI 6727) is a highly potent Plk1 inhibitor with IC50 of 0.87 nM in a cell-free assay. It shows 6- and 65-fold greater selectivity against Plk2 and Plk3. |
1608125-21-8 |
AMG319 |
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AMG319 is a potent and selective PI3Kδ inhibitor with IC50 of 18 nM, >47-fold selectivity over other PI3Ks |
1620576-64-8 |
AZD8835 |
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AZD8835 is an effective and selective PI3K inhibitors of PI3K and δ α, the IC50 values were 5.7 and 6.2 nM nM, selective than the PI3K-beta (IC50 to 431 nM) and PI3K gamma (I... |
1627494-13-6 |
AZD8186 |
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AZD8186 is a potent and selective inhibitor of PI3Kβ and PI3Kδ with IC50 of 4 nM and 12 nM, respectively. |
1276553-09-3 |
PF-4989216 |
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PF-4989216 is a potent and selective PI3K inhibitor with IC50 of 2 nM, 142 nM, 65 nM, 1 nM, and 110 nM for p110α, p110β, p110γ, p110δ, and VPS34, respectively. |
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